CLASSIFICATION: GROWTH HORMONE SECRETAGOGUE
ACTIVE SUBSTANCE: EXAMORELIN (HEXARELIN)
FORM: LYOPHILIZED POWDER (2 ML VIAL x 5 MG)
ACTIVE HALF-LIFE: APPROX. 55 MINUTES
DOSAGE: 100–200 MCG 1–2X DAILY (RESEARCH USE)
ACNE: UNLIKELY
WATER RETENTION: MILD
HIGH BLOOD PRESSURE (HBP): UNLIKELY
HEPATOTOXICITY: NONE
AROMATIZATION: NO
MANUFACTURER: PEPTIDE HUBS
Hexarelin (also known as Examorelin) is a synthetic growth hormone-releasing peptide (GHRP) with one of the strongest GH pulse responses in its class. It is frequently used in research examining muscle development, recovery, pituitary responsiveness, and cardiac tissue regeneration. Peptide Hubs offers Hexarelin in a 5 mg lyophilized vial—ideal for sustained protocols in endocrine and anti-aging research.
Hexarelin binds to the ghrelin receptor (GHS-R1a) and acts directly on the hypothalamus and pituitary to stimulate endogenous GH release. Compared to GHRP-2 or GHRP-6, Hexarelin induces a stronger, more sustained GH pulse without significantly raising appetite. In addition to its GH effects, animal models have shown potential cardioprotective properties. For peer-reviewed data, refer to this NIH article on Hexarelin and cardiac function.
Hexarelin is often co-administered with CJC-1295 DAC to prolong GH activity, or AOD 9604 in metabolic optimization research. Researchers also stack it with B7-33 for potential synergy in cardiac fibrosis reduction models.
Hexarelin is often combined with synergistic peptides in preclinical settings:
Hexarelin is for research use only and is not FDA-approved for human or veterinary use. It exhibits no aromatization, no hepatic stress, and minimal risk of appetite stimulation or prolactin elevation. For updates on clinical research, consult ClinicalTrials.gov.
Hexarelin is studied for its strong GH pulse, support in muscle regeneration, metabolic performance, and cardiac repair in preclinical models.
Yes. Hexarelin produces a stronger and more prolonged GH release compared to GHRP-2 and GHRP-6, with fewer hunger-related side effects.
Unlike GHRP-6, Hexarelin has minimal impact on appetite, making it suitable for studies focusing purely on GH secretion and tissue repair.
No. Hexarelin is not FDA-approved and is sold strictly for laboratory research purposes only.
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CLASSIFICATION: GROWTH HORMONE SECRETAGOGUE (GHS)
ACTIVE SUBSTANCE: EXAMORELIN
FORM: 2 ML VIAL x 5 MG (LYOPHILIZED POWDER)
ACTIVE HALF-LIFE: APPROX. 60–90 MINUTES
DOSAGE: 100–200 MCG, 2–3 TIMES DAILY
ACNE: RARE
WATER RETENTION: MILD
HBR: NO
HEPATOTOXICITY: NO
AROMATIZATION: NO
MANUFACTURER: DRAGON PHARMA
LABORATORY TESTED: VIEW LAB RESULTS
CLASSIFICATION: RECOMBINANT HUMAN GROWTH HORMONE (rHGH)
ACTIVE SUBSTANCE: SOMATROPIN
FORM: 1 PRE-FILLED PEN x 36 IU (12 MG)
ACTIVE HALF-LIFE: ~3.5 HOURS (SUBQ)
DOSAGE: 1–4 IU/DAY FOR ANTI-AGING; 4–8 IU/DAY FOR FAT LOSS OR PERFORMANCE
WATER RETENTION: POSSIBLE (DOSE DEPENDENT)
HEPATOTOXICITY: NONE
AROMATIZATION: NO
MANUFACTURER: PFIZER
CLASSIFICATION: RECOMBINANT HUMAN GROWTH HORMONE (r-hGH)
ACTIVE SUBSTANCE: SOMATROPIN (R-HGH)
FORM: 1 CARTRIDGE x 15 MG
ACTIVE HALF-LIFE: ~2–3 HOURS
DOSAGE: MEN 4-10 IU/DAY
ACNE: POSSIBLE
WATER RETENTION: POSSIBLE
HIGH BLOOD PRESSURE (HBP): MAY INCREASE VIA FLUID RETENTION
HEPATOTOXICITY: NONE TYPICAL
AROMATIZATION: NONE
MANUFACTURER: NOVO NORDISK
CLASSIFICATION: GONADOTROPIN (LH RECEPTOR AGONIST)
ACTIVE SUBSTANCE: HUMAN CHORIONIC GONADOTROPIN
FORM: 1 LYOPHILIZED VIAL x 5000 IU + PROVIDED SOLVENT
ACTIVE HALF-LIFE: ~24–36 HOURS
DOSAGE: MEN 500-1000 IU
ACNE: POSSIBLE
WATER RETENTION: POSSIBLE
HIGH BLOOD PRESSURE (HBP): MONITOR IF AT CV RISK
HEPATOTOXICITY: NONE TYPICAL
AROMATIZATION: INDIRECT
MANUFACTURER: IBSA
CLASSIFICATION: PEPTIDE HORMONE / HCG
ACTIVE SUBSTANCE: HUMAN CHORIONIC GONADOTROPIN
FORM: 1 ML AMP x 5000 IU
ACTIVE HALF-LIFE: ~3–6 DAYS
DOSAGE: 250–1000 IU 2–3x/WEEK (ON-CYCLE or PCT)
ACNE: POSSIBLE
WATER RETENTION: MODERATE
HIGH BLOOD PRESSURE (HBP): UNLIKELY
HEPATOTOXICITY: NONE
AROMATIZATION: INDIRECTLY ELEVATES ESTROGEN
MANUFACTURER: SUN PHARMA